Adrenoblockers ama adrenolytics waa daroogo si gaabis ah ama xannibaya marinka dareemayaasha, i.e. waxay "damiyaan" kuwa soo dhaweeyaha ee ku yaala derbiyada xididdada dhiigga iyo wadnaha, taas oo ka jawaabta adrenaline iyo norepinephrine. Liiska daawooyinka-adrenoblockers wuxuu noqonayaa mid aad u ballaaran sanad walba. Aynu isku dayno inaan ogaano nooca adrenolytics ee jira, iyo sidoo kale waxa dabeecadaha ay wax ku ool yihiin.
Maxay yihiin mukhadaraadka iyo daawooyinka beta-adrenoblockers?
Noocyada ugu waaweyn ee adrenoblockers waa:
- alfa-blockers;
- beta-blockers.
Iyada oo ku xiran nooca adrenolytics wuxuu saameeyaa soo dhaweeye mid ka mid ah labada nooc.
Adrenoblockers kala duwan ayaa leh qaab kala duwan. Sidaas awgeed adrenolytics ayaa lagu soo saarey foomka:
- Kiniiniyada;
- dhalada oo leh xalka cirbadaha;
- dhibcood.
Xayiraadaha Alpha
Alpha-adrenoblockers ee jirka ku dhaqma sida soo socota:
- ballaadhiyaan xididada yar, iyadoo yareyneysa culeyska wadnaha;
- yaree cadaadiska wadnaha, hoos u dhigista iska caabinta dhuumaha xididdada dhiigga iyo culeyska muruqyada wadnaha;
- hagaajinta wareegga dhiigga;
- yaree cadaadiska wareegga yar ee wareegga wareegga wareegga;
- kolestaroolka hoose;
- yareeyo xaddiga gulukooska ee dhiigga.
Kooxda xayiraadaha alfa-receptor waxaa ka mid ah daroogooyinka loo isticmaalo dariiqooyinka soo socda:
- dhiig-karka;
- xanuunka dhanjafka ;
- endadoitis;
- istiraashka maraakiibta retina.
Alpha-adrenoblockers ayaa si guul leh loogu isticmaalaa daaweynta adag ee prostatitis ee ragga.
Xasaasiyadaha isticmaalka alfa-blockers waa cudurada:
- qalalaasaha araga;
- atherosclerosis;
- cudurka miyir-qaadiga;
- xayeysiin keli ah ama "hepatic".
Liistada diyaargarowga caanka ah ee alfa-blockers:
- Dihydroergotoksin;
- Urapidil;
- Nicergoline;
- Fentolamine;
- Pyrroxane;
- Tropafen;
- Prazosin hydrochloride;
- Butyroxane.
Macluumaadka! Markii hore, daroogooyinka laga helay liiska xayiraadaha ayaa loo adeegsan jiray wadnaha oo dhan daaweynta dhammaan bukaannada iyada oo aan ka reeban, laakiin natiijada baadhitaan caafimaad ayaa la ogaaday in mararka qaarkood codsigoodu uu keeni karo wadne qabad.
Beta-aqbalaha xayiraadaha
Maamulka dawooyinka beta-blocker ayaa keenaya saameynta soo socota:
- hoos u dhigida garaaca wadnaha;
- cadaadiska dhiigga;
- caabbinta unugyada muruqyada wadnaha si loogu helo gaajo oksijiin ah is-kicinta;
- waxay hagaajineysaa codka maraakiibta dhiigga;
- sameynta thrombocytes waa la joojiyaa;
- waxay kordhisaa socodka oksijiinka unugyada jirka;
- shaqada qalliinnada gudaha iyo qanjirada qarsoodiga ayaa xasillan.
Tilmaamaha loogu talagalay isticmaalka mukhaadaraadka liiska kudhaca β-blockers waa cudurada sida:
- glaucoma;
- dhiig-karka;
- pectoris angina;
- xannuunka wadnaha;
- cudurka miyir-qaadiga;
- Wadnaha wadnaha;
- thyrotoxicosis ;
- qaadashada wadnaha.
Waxyaabaha ka soo horjeeda isticmaalka daroogooyinka noocaan ah waa dhowr cudur, oo ay ka mid yihiin:
- diabetes mellitus;
- neefta neefta;
- COPD (cudurada joogtada ah ee joogtada ah);
- joojinta atherosclerosis.
Liiska liiska beta-blockers ee jiilka cusub, daroogooyinka:
- Cormum;
- Anaprilin (Propranolol);
- Metoprolol;
- Bisoprolol (Concor);
- Nabilet (Nebivolol);
- Betaxolol (Lokren);
- Aptin;
- Betazprin;
- Esmolol et al.
Muhiim! Inkastoo inkastoo daroogooyinka qaarkood-adrenoblockers laga iibsan karo farmashiyo la'aanteed rijeeto, laakiin waa in loo isticmaalo sida waafaqsan rijeetada takhtarka, sababtoo ah waxyeello culus ayaa la heli karaa meeshii laga heli lahaa daaweyn wax ku ool ah.
Adrenoblockers oo isku dhafan
Waxaa jira koox gaar ah oo daroogo ah oo isu muujiya isla markiiba sida daawooyinka alfa adrenolytics iyo daawooyinka beta-adrenolytic. Kuwani waa adrenoblockers, sida:
- Labeetool;
- Procodolol.